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Naquotinib mesylate (ASP8273 mesylate) is an orally available, mutant-selective and irreversible EGFR inhibitor; with IC50s of 8-33 nM toward EGFR mutants and 230 nM for EGFR.
| Molecular Weight | 658.81 |
| CAS Number | 1448237-05-5 |
| Solubility (25°C) | DMSO 12.5 mg/mL |
| Storage | 2-8°C, dry, sealed |
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