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MRS 1477 

Cat. No. M29264

All AbMole products are for research use only, cannot be used for human consumption.

MRS 1477  Structure

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Quality Control & Documentation
Biological Activity

MRS 1477, a dihydropyridine derivative, is a positive allosteric modulator of TRPV1 in the presence of capsaicin. MRS 1477 itself does not induce apoptosis, but the co-existence of MRS 1477 and capsaicin can induce apoptosis.

Chemical Information
Molecular Weight 389.51
Formula C21H27NO4S
CAS Number 212200-21-0
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] Luka Flegar, et al. Eur J Nucl Med Mol Imaging. Adoption of Lutetium-177 PSMA radioligand therapy for metastatic castration resistant prostate cancer: a total population analysis in Germany from 2016 to 2020

[2] Luka Flegar, et al. World J Urol. Treatment trends for muscle-invasive bladder cancer in Germany from 2006 to 2019

[3] Taous-Meriem Laleg-Kirati, et al. NMR Biomed. Spectral data de-noising using semi-classical signal analysis: application to localized MRS

[4] Ruiqin Zhang, et al. Int J Clin Exp Med. Prevalence of multidrug resistant Gram-positive cocci in a Chinese hospital over an 8-year period

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Keywords: MRS 1477  supplier, TRP Channel, inhibitors, activators

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