Free shipping on all orders over $ 500

ML-290

Cat. No. M45103

All AbMole products are for research use only, cannot be used for human consumption.

ML-290 Structure

Price and Availability

For this product's availability, delivery time and price, please email [email protected] directly or click the "Inquiry Now" button below.

Quality Control & Documentation
Biological Activity

ML-290 is a first-in-class, potent relaxin/glucagon-like peptide receptor (RXFP1) agonist and anti-fibrotic gene activator with an EC50 value of 94 nM.

Chemical Information
Molecular Weight 506.49
Formula C24H21F3N2O5S
CAS Number 1482500-76-4
Form Solid
Solubility (25°C) DMSO >100 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Sai Nivedita Krishnan, et al. Biochim Biophys Acta Mol Basis Dis. Human C1q Tumor Necrosis Factor 8 (CTRP8) defines a novel tryptase+ mast cell subpopulation in the prostate cancer microenvironment

[2] Kenneth J Wilson, et al. Eur J Med Chem. Optimization of the first small-molecule relaxin/insulin-like family peptide receptor (RXFP1) agonists: Activation results in an antifibrotic gene expression profile

Related Products
D-Allulose

D-Allulose (D-Psicose) is an ultralow-energy monosaccharide sugar. It is a C-3 epimer of D-fructose, and is present in small quantities in agricultural products and commercially-prepared carbohydrate complexes.
N,N-Dimethyltrifluoromethanesulfonamide

N,N-Dimethyltrifluoromethanesulfonamide (DMTMSA) is a trifluoromethanesulfonamide solvent.
Lucicebtide

Lucicebtide is a peptide antagonist of the transcription factor C/EBPβ, a key activator of the transcriptional program in immunosuppressive macrophages. Lucicebtide shows highly potent inhibition against C/EBPB-ATF5 association with IC50 of 24.6 nM in a competitive ELISA assay.
Eloralintide

Eloralintide (LY 3841136) is an AMYR agonist.
Gadoteric acid

Gadoteric acid is a macrocyclic, paramagnetic, gadolinium-based contrast agent that can be used for magnetic resonance imaging (MRI) of the brain, spine, and related tissues. Gadoteric acid is able to detect and visualize areas of blood-brain barrier disruption and abnormal vascular distribution.
  Catalog
Abmole Inhibitor Catalog




Keywords: ML-290 supplier, inhibitors, activators

All AbMole products are for research use only, cannot be used for human consumption or veterinary use. We do not provide products or services to individuals. Please comply with the intended use and do not use AbMole products for any other purpose.


 
Get to Know Us
Customer Support
Resources
Contact Us

Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2024 AbMole BioScience. All Rights Reserved.