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ML-290

Cat. No. M45103

All AbMole products are for research use only, cannot be used for human consumption.

ML-290 Structure

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Quality Control & Documentation
Biological Activity

ML-290 is a first-in-class, potent relaxin/glucagon-like peptide receptor (RXFP1) agonist and anti-fibrotic gene activator with an EC50 value of 94 nM.

Chemical Information
Molecular Weight 506.49
Formula C24H21F3N2O5S
CAS Number 1482500-76-4
Form Solid
Solubility (25°C) DMSO >100 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Sai Nivedita Krishnan, et al. Biochim Biophys Acta Mol Basis Dis. Human C1q Tumor Necrosis Factor 8 (CTRP8) defines a novel tryptase+ mast cell subpopulation in the prostate cancer microenvironment

[2] Kenneth J Wilson, et al. Eur J Med Chem. Optimization of the first small-molecule relaxin/insulin-like family peptide receptor (RXFP1) agonists: Activation results in an antifibrotic gene expression profile

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Keywords: ML-290 supplier, inhibitors, activators

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