Free shipping on all orders over $ 500

Metergoline

Cat. No. M7924

All AbMole products are for research use only, cannot be used for human consumption.

Metergoline Structure
Size Price Availability Quantity
10mg USD 60  USD60 In stock
Free Delivery on orders over USD 500 Bulk Inquiry?

Quality Control & Documentation
Biological Activity

Antagonist at 5-HT1, 5-HT2, and 5-HT7 serotonin receptors; analgesic; antipyretic.

Chemical Information
Molecular Weight 403.52
Formula C25H29N3O2
CAS Number 17692-51-2
Solubility (25°C) 0.1 M HCl: 1.4 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Hyoung-Woo Bai, et al. Molecular basis involved in the blocking effect of antidepressant metergoline on C-type inactivation of Kv1.4 channel

[2] Jun-Ho Lee, et al. Metergoline inhibits the neuronal Nav1.2 voltage-dependent Na(+) channels expressed in Xenopus oocytes

[3] Kai Kang, et al. Metergoline-induced cell death in Candida krusei

[4] A Caballero Sr, et al. Metergoline as a lactation inhibitor

[5] C Ferrari, et al. Endocrine profile and therapeutic employment of a new prolactin-lowering drug, metergoline

Related Products
GAPDH-IN-1

GAPDH-IN-1 (GAPDH Inhibitor Compound F8) is a covalent inhibitor of GAPDH (IC50 = 39.31 µM). It viability of, and glucose metabolism in, HEK293 cells in a concentration-dependent manner.

O-acetylcamptothecin

O-acetylcamptothecin is a derivative of camptothecin, a naturally occurring alkaloid extracted from the bark of the Chinese tree Camptotheca acuminata. Camptothecin and its derivatives are primarily known for their potent anticancer properties, particularly through their action as inhibitors of topoisomerase I, an enzyme critical for DNA replication and transcription.

10-hydroxystearic acid

10-hydroxystearic acid is a hydroxy fatty acid.

SB-T-1214

SB-T-1214 is a new-generation taxoid. SB-T-1214 possesses significant activity against colon cancer spheroids induced by and enriched with drug resistant tumorigenic CD133high/CD44high cells and efficiently inhibited expression of the majority of stem cell-related genes.

NG-497

NG-497 is a selective human adipose triglyceride lipase (ATGL) inhibitor that targets the enzymatically active patatin-like domain of human ATGL.

  Catalog
Abmole Inhibitor Catalog




Keywords: Metergoline supplier, inhibitors, activators

All AbMole products are for research use only, cannot be used for human consumption or veterinary use. We do not provide products or services to individuals. Please comply with the intended use and do not use AbMole products for any other purpose.



Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2024 AbMole BioScience. All Rights Reserved.