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Levocabastine

Cat. No. M30621

All AbMole products are for research use only, cannot be used for human consumption.

Levocabastine Structure
Synonym:

R 50547

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Quality Control & Documentation
Biological Activity

Levocabastine (R 50547) is a potent and selective histamine H1-receptor antagonist. Levocabastine hydrochloride is also a selective, high affinity neurotensin receptor subtype 2 (NTR2) antagonist, with a Ki of 17 nM for mNTR2. Levocabastine can act as a VLA-4 antagonist, interferes with conjunctival eosinophil infiltration in allergic conjunctivitis (AC).

Chemical Information
Molecular Weight 420.52
Formula C26H29FN2O2
CAS Number 79516-68-0
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] No authors listed. Levocabastine

[2] S Noble, et al. Drugs. Levocabastine. An update of its pharmacology, clinical efficacy and tolerability in the topical treatment of allergic rhinitis and conjunctivitis

[3] K L Dechant, et al. Drugs. Levocabastine. A review of its pharmacological properties and therapeutic potential as a topical antihistamine in allergic rhinitis and conjunctivitis

[4] M M Janssens, et al. Clin Exp Allergy. Levocabastine: an effective topical treatment of allergic rhinoconjunctivitis

[5] M M Janssens. Rhinol Suppl. Levocabastine: a new topical approach for the treatment of paediatric allergic rhinoconjunctivitis

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Keywords: Levocabastine, R 50547 supplier, Histamine Receptor, inhibitors, activators

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