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KSK67

Cat. No. M42695

All AbMole products are for research use only, cannot be used for human consumption.

KSK67 Structure

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Quality Control & Documentation
Biological Activity

KSK67 is a high-affinity dual sigma-2 and histamine H3 receptor antagonist, with Kis of 3.2, 1531, 101 nM for H3 receptor, sigma-1, sigma-2 receptor respectively.

Chemical Information
Molecular Weight 365.47
Formula C22H27N3O2
CAS Number 2566715-93-1
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Katarzyna Szczepańska et al. J Med Chem. Dual Piperidine-Based Histamine H3 and Sigma-1 Receptor Ligands in the Treatment of Nociceptive and Neuropathic Pain

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Keywords: KSK67 supplier, Sigma Receptor, inhibitors, activators

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