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JNJ-1013

Cat. No. M41291

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JNJ-1013 Structure

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Quality Control & Documentation
Biological Activity

JNJ-1013 is a potent and selective IRAK1 degrader with an IC50s of 72, 443, 1071 nM for IRAK1, IRAK4, VHL FP respectively.

Chemical Information
Molecular Weight 878.05
Formula C46H55N9O7S
CAS Number 2597343-08-1
Form Solid
Solubility (25°C) DMSO 20 mg/mL (ultrasonic and warming)
Storage 4°C, protect from light
References

[1] Liqiang Fu et al. J Med Chem. Discovery of Highly Potent and Selective IRAK1 Degraders to Probe Scaffolding Functions of IRAK1 in ABC DLBCL

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  Catalog
Abmole Inhibitor Catalog




Keywords: JNJ-1013 supplier, IRAK, inhibitors, activators

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