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Itraconazole

Cat. No. M5719

All AbMole products are for research use only, cannot be used for human consumption.

Itraconazole Structure
Synonym:

R 51211

Size Price Availability Quantity
100mg USD 50  USD50 In stock
500mg USD 120  USD120 In stock
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Quality Control & Documentation
Biological Activity

Itraconazole is a relatively potent inhibitor of CYP3A4 with IC50 of 6.1 nM, used as a triazole antifungal agent.

Chemical Information
Molecular Weight 705.65
Formula C35H38Cl2N8O4
CAS Number 84625-61-6
Form Solid
Solubility (25°C) 7 mg/mL warmed in DMSO
Storage 2-8°C, protect from light
References

[1] Abuhelwa AY, et al. Antimicrob Agents Chemother. Population pharmacokinetic modeling of itraconazole and hydroxyitraconazole for oral SUBA-itraconazole and sporanox capsule formulations in healthy subjects in fed and fasted states.

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Keywords: Itraconazole, R 51211 supplier, Antibiotic, inhibitors, activators

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