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Inupadenant

Cat. No. M29428

All AbMole products are for research use only, cannot be used for human consumption.

Inupadenant Structure
Synonym:

EOS-850

Price and Availability

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Quality Control & Documentation
Biological Activity

Inupadenant is an orally active, highly selective A2A receptor antagonist. Inupadenant is not brain-penetrant. Inupadenant has potent anti-tumor activity.

Chemical Information
Molecular Weight 604.65
Formula C25H26F2N8O4S2
CAS Number 2246607-08-7
Form Solid
Solubility (25°C) DMSO 40 mg/mL (ultrasonic and warming and adjust pH to 4 with HCl and heat to 60°C)
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] S-A Im, et al. ESMO Open. Pan-Asian adapted ESMO Clinical Practice Guidelines for the diagnosis, staging and treatment of patients with metastatic breast cancer

[2] F Cortiula, et al. Ann Oncol. Immunotherapy in unresectable stage III non-small-cell lung cancer: state of the art and novel therapeutic approaches

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  Catalog
Abmole Inhibitor Catalog




Keywords: Inupadenant, EOS-850 supplier, Adenosine Receptor, inhibitors, activators

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