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GSK726701A

Cat. No. M10827

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GSK726701A  Structure

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Quality Control & Documentation
Biological Activity

GSK726701A is a partial agonist of prostaglandin E2 receptor 4 (EP4),pEC50is 7.4.

Chemical Information
Molecular Weight 423.43
Formula C24H22FNO5
CAS Number 945721-87-9
Solubility (25°C) DMSO ≥ 20 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Mark P Healy, et al. Bioorg Med Chem Lett. Discovery of {4-[4,9-bis(ethyloxy)-1-oxo-1,3-dihydro-2H-benzo[f]isoindol-2-yl]-2-fluorophenyl}acetic acid (GSK726701A), a novel EP 4 receptor partial agonist for the treatment of pain

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  Catalog
Abmole Inhibitor Catalog




Keywords: GSK726701A supplier, Prostaglandin Receptor, inhibitors, activators

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