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GSK3395879 

Cat. No. M29363

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GSK3395879  Structure

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Quality Control & Documentation
Biological Activity

GSK3395879 is a selective and orally bioavailable transient receptor potential vanilloid-4 (TRPV4) antagonist with an IC50 of 1 nM for hTRPV4.

Chemical Information
Molecular Weight 485.41
Formula C20H15F4N3O5S
CAS Number 2215852-91-6
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] Edward J Brnardic, et al. J Med Chem. Discovery of Pyrrolidine Sulfonamides as Selective and Orally Bioavailable Antagonists of Transient Receptor Potential Vanilloid-4 (TRPV4)

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  Catalog
Abmole Inhibitor Catalog




Keywords: GSK3395879  supplier, TRP Channel, inhibitors, activators

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