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GNE-9815

Cat. No. M21135

All AbMole products are for research use only, cannot be used for human consumption.

GNE-9815 Structure

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Quality Control & Documentation
Biological Activity

GNE-9815 is one of the most selective kinase inhibitors of RAF, targeting KRAS mutant cancers by combination of drugs.

Chemical Information
Molecular Weight 455.48
Formula C26H22FN5O2
CAS Number 2729996-45-4
Solubility (25°C) DMSO : 50 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Malcolm P Huestis, et al. ACS Med Chem Lett. Targeting KRAS Mutant Cancers via Combination Treatment: Discovery of a Pyridopyridazinone pan-RAF Kinase Inhibitor

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  Catalog
Abmole Inhibitor Catalog




Keywords: GNE-9815 supplier, Raf, inhibitors, activators

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