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GLPG3970

Cat. No. M40967

All AbMole products are for research use only, cannot be used for human consumption.

GLPG3970 Structure

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Quality Control & Documentation
Biological Activity

GLPG3970 is a first-in-class salt-inducible kinase SIK2/SIK3 inhibitor for studies related to inflammatory and autoimmune diseases such as psoriasis.

Chemical Information
Molecular Weight 504.50
Formula C25H27F3N4O4
CAS Number 2403733-82-2
Form Solid
Solubility (25°C) DMSO 90 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Wei Zhu et al. Bioorg Med Chem. Discovery of novel and selective SIK2 inhibitors by the application of AlphaFold structures and generative models

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  Catalog
Abmole Inhibitor Catalog




Keywords: GLPG3970 supplier, Salt-inducible Kinase, inhibitors, activators

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