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GFB-887

Cat. No. M43953

All AbMole products are for research use only, cannot be used for human consumption.

GFB-887 Structure
Synonym:

KAR-2618

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Quality Control & Documentation
Biological Activity

GFB-887 is an inhibitor of transient receptor potential channels 4 and 5 (TRPC4/5) and can be used in studies related to anxiety disorders.

Chemical Information
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Amy D Westerling-Bui, et al. Sci Adv. Transplanted organoids empower human preclinical assessment of drug candidate for the clinic

[2] Liron Walsh, et al. Kidney Int Rep. Safety and Efficacy of GFB-887, a TRPC5 Channel Inhibitor, in Patients With Focal Segmental Glomerulosclerosis, Treatment-Resistant Minimal Change Disease, or Diabetic Nephropathy: TRACTION-2 Trial Design

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Keywords: GFB-887, KAR-2618 supplier, TRP Channel, inhibitors, activators

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