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GAK inhibitor 49

Cat. No. M58414

All AbMole products are for research use only, cannot be used for human consumption.

GAK inhibitor 49 Structure
Size Price Availability Quantity
1mg USD 120  USD120 In stock
5mg USD 260  USD260 In stock
10mg USD 400  USD400 In stock
25mg USD 700  USD700 In stock
50mg USD 1000  USD1000 In stock
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Quality Control & Documentation
Biological Activity

GAK inhibitor 49 is a potent, ATP-competitive and highly selective cyclin G associated kinase (GAK) inhibitor with a Ki of 0.54 nM and a cell IC50 of 56 nM. 

Chemical Information
Molecular Weight 370.4
Formula C20H22N2O5
CAS Number 319492-82-5
Solubility (25°C) DMSO 37 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
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Keywords: GAK inhibitor 49 supplier, inhibitors, activators

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