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Enprofylline

Cat. No. M30061

All AbMole products are for research use only, cannot be used for human consumption.

Enprofylline Structure

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Quality Control & Documentation
Biological Activity

Enprofylline acts as a selective and competitive A2B receptor antagonist with the Ki of 7 μM. Enprofylline also acts as a phosphodiesterase inhibitor. Enprofylline can be used for the research of asthma, chronic obstructive pulmonary disease.

Chemical Information
Molecular Weight 194.19
Formula C8H10N4O2
CAS Number 41078-02-8
Form Solid
Solubility (25°C) DMSO 62.5 mg/mL (ultrasonic)
Storage 4°C, protect from light
References

[1] K R Chapman, et al. Chest. Long-term xanthine therapy of asthma. Enprofylline and theophylline compared. International Enprofylline Study Group

[2] M Esquivel, et al. Clin Pharmacol Ther. Cardiovascular effects of enprofylline and theophylline

[3] B J Chapman, et al. Br J Dis Chest. Enprofylline in chronic asthma

[4] C G Persson, et al. Life Sci. Effects of enprofylline and theophylline may show the role of adenosine

[5] I Muraoka, et al. Drug Metab Dispos. Pharmacokinetics and renal handling of enprofylline in pregnant rats

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Keywords: Enprofylline supplier, Adenosine Receptor, inhibitors, activators

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