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EHT 1610

Cat. No. M14888

All AbMole products are for research use only, cannot be used for human consumption.

EHT 1610 Structure

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Quality Control & Documentation
Biological Activity

EHT 1610 is a strong inhibitor of DYRK’s family kinases, with IC50s of 0.36, 0.59 nM for DYRK1A and DYRK1B, respectively.

<span style='color:#ff0000;'><strong>*The compound is unstable in solutions, freshly prepared is recommended</strong></span>


Chemical Information
Molecular Weight 383.4
CAS Number 1425945-60-3
Solubility (25°C) DMSO 5 mg/mL
Storage -20°C, protect from light, sealed
References

[1] Apirat Chaikuad, et al. An Unusual Binding Model of the Methyl 9-Anilinothiazolo[5,4-f] quinazoline-2-carbimidates (EHT 1610 and EHT 5372) Confers High Selectivity for Dual-Specificity Tyrosine Phosphorylation-Regulated Kinases

[2] Alicia Foucourt, et al. Design and synthesis of thiazolo[5,4-f]quinazolines as DYRK1A inhibitors, part II

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  Catalog
Abmole Inhibitor Catalog




Keywords: EHT 1610 supplier, inhibitors, activators

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