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EEDi-5273

Cat. No. M11355

All AbMole products are for research use only, cannot be used for human consumption.

EEDi-5273  Structure

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Quality Control & Documentation
Biological Activity

Eedi-5273 is a potent and orally effective EED inhibitor (IC50 = 0.2 nM) that can achieve complete and sustained tumor regression.

Chemical Information
Molecular Weight 526.49
Formula C26H22F4N6O2
CAS Number 2585648-55-9
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Rohan Kalyan Rej, et al. J Med Chem. Discovery of EEDi-5273 as an Exceptionally Potent and Orally Efficacious EED Inhibitor Capable of Achieving Complete and Persistent Tumor Regression

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  Catalog
Abmole Inhibitor Catalog




Keywords: EEDi-5273 supplier, PRC2/EED, inhibitors, activators

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