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Delphinidin chloride

Cat. No. M10417
Delphinidin chloride Structure
Synonym:

delfinidolchloride

Size Price Availability Quantity
1mg USD 198  USD220 In stock
10mg USD 594  USD660 In stock
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Quality Control
  • Current batch:
  • Purity >98%
  • COA
  • MSDS
Biological Activity

Delphinidin (chloride) is an anthocyanidin, a natural plant pigment which can modulate JAK/STAT3 and MAPKinase signaling to induce apoptosis in HCT116 cells. Delphinidin chloride shows endothelium-dependent vasorelaxation. It also inhibits signaling through epithelial growth factor receptors, suppressing the expression of estrogen receptor α and inducing both apoptosis and autophagy at a dose of 1-40 μM.

Conversion of different model animals based on BSA (Value based on data from FDA Draft Guidelines)
Species Mouse Rat Rabbit Guinea pig Hamster Dog
Weight (kg) 0.02 0.15 1.8 0.4 0.08 10
Body Surface Area (m2) 0.007 0.025 0.15 0.05 0.02 0.5
Km factor 3 6 12 8 5 20
Animal A (mg/kg) = Animal B (mg/kg) multiplied by  Animal B Km
Animal A Km

For example, to modify the dose of Compound A used for a mouse (20 mg/kg) to a dose based on the BSA for a rat, multiply 20 mg/kg by the Km factor for a mouse and then divide by the Km factor for a rat. This calculation results in a rat equivalent dose for Compound A of 10 mg/kg.

Chemical Information
Molecular Weight 338.7
Formula C15H11ClO7
CAS Number 528-53-0
Purity >98%
Solubility DMSO 50 mg/mL
Storage 2-8°C, protect from light, sealed
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  Catalog
Abmole Inhibitor Catalog 2017




Keywords: Delphinidin chloride, delfinidolchloride supplier, JAK, inhibitors

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