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Debrisoquin hemisulfate

Cat. No. M42350

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Debrisoquin hemisulfate Structure

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Quality Control & Documentation
Biological Activity

Debrisoquin (Isocaramidine) hemisulfate is a TMPRSS2 inhibitors that inhibits SARS-CoV-2 entry into human lung cell line by a TMPRSS2-depedent manner, with an IC50 of 22μM.

Chemical Information
Molecular Weight 224.27
Formula C10H13N3.1/2H2O4S
CAS Number 581-88-4
Form Solid
Solubility (25°C) Water 10 mg/mL (ultrasonic and warming)
Storage Powder -20°C 3 years
References

[1] Yueying Zhen et al. Drug Metab Dispos. 3,4-Dehydrodebrisoquine, a novel debrisoquine metabolite formed from 4-hydroxydebrisoquine that affects the CYP2D6 metabolic ratio

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Keywords: Debrisoquin hemisulfate supplier, Metabolite/Endogenous Metabolite, inhibitors, activators

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