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Contezolid

Cat. No. M27802

All AbMole products are for research use only, cannot be used for human consumption.

Contezolid Structure
Synonym:

MRX-I

Size Price Availability Quantity
1mg USD 300  USD300 In stock
5mg USD 700  USD700 In stock
10mg USD 1000  USD1000 In stock
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Quality Control & Documentation
Biological Activity

Contezolid (MRX-I), a new and orally active oxazolidinone, is an antibiotic in study for complicated skin and soft tissue infections (cSSTI) caused by resistant Gram-positive bacteria. Contezolid (MRX-I) markedly reduces potential for myelosuppression and monoamine oxidase inhibition (MAOI).

Chemical Information
Molecular Weight 408.33
Formula C18H15F3N4O4
CAS Number 1112968-42-9
Form Solid
Solubility (25°C) DMSO 120 mg/mL (ultrasonic)
Storage 4°C, protect from light, dry, sealed
References

[1] Grace Kaul, et al. Drugs Today (Barc). Contezolid in complicated skin and soft tissue infection

[2] Min Yang, et al. Drug Discov Ther. Prospects of contezolid (MRX-I) against multidrυg-resistant tuberculosis and extensively drυg-resistant tuberculosis

[3] Sheridan M Hoy. Drugs. Correction to: Contezolid: First Approval

[4] Qi Guo, et al. Antimicrob Agents Chemother. A Novel Oxazolidinone, Contezolid (MRX-I), Expresses Anti-Mycobacterium abscessus Activity In Vitro

[5] Sheridan M Hoy. Drugs. Contezolid: First Approval

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Keywords: Contezolid, MRX-I supplier, Antibiotic, inhibitors, activators

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