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Cetrorelix Acetate (SB-75 acetate) is a potent gonadotropin-releasing hormone (GnRH) receptor antagonist with an IC50 of 1.21 nM. Cetrorelix Acetate inhibits growth of ES-2 cell line at 1000 ng/ml. Cetrorelix Acetate has comparable antiproliferative effects as GnRH-I agonists indicating that the dichotomy of GnRH-I agonists and antagonists might not apply to the GnRH-I system in cancer cells.
Sequence：Ac-D2Nal-D4Cpa-D3Pal-Ser-Tyr-DCit-Leu-Arg-Pro-DAla-NH2
| Molecular Weight | 1491.09 |
| Formula | C72H96ClN17O16 |
| CAS Number | 145672-81-7 |
| Solubility (25°C) | Water 2 mg/mL DMSO 30 mg/mL |
| Storage | -20°C, protect from light, dry, sealed |
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