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Centanafadine hydrochloride

Cat. No. M43921

All AbMole products are for research use only, cannot be used for human consumption.

Centanafadine hydrochloride Structure
Synonym:

EB-1020 hydrochloride

Size Price Availability Quantity
5mg USD 150  USD150 In stock
10mg USD 240  USD240 In stock
25mg USD 480  USD480 In stock
50mg USD 750  USD750 In stock
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Quality Control & Documentation
Biological Activity

Centanafadine hydrochloride is a potential first-in-class norepinephrine (NE), dopamine (DA), and 5-hydroxytryptamine (5-HT) reuptake inhibitor (NDSRI) with IC50 values of 6 nM, 38 nM, and 83 nM, respectively. It can be used in studies related to attention-deficit/hyperactivity disorder (ADHD).

Chemical Information
Molecular Weight 245.75
Formula C15H16ClN
CAS Number 923981-14-0
Form Solid
Solubility (25°C) DMSO >100 mg/mL
Storage 4°C, dry, sealed
References

[1] Fatuma Nageye, et al. Expert Rev Neurother. Beyond stimulants: a systematic review of randomised controlled trials assessing novel compounds for ADHD

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Keywords: Centanafadine hydrochloride, EB-1020 hydrochloride supplier, Serotonin Transporter, inhibitors, activators

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