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BRL 50481

Cat. No. M6533

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BRL 50481 Structure
Size Price Availability Quantity
5mg USD 60  USD60 In stock
10mg USD 80  USD80 In stock
25mg USD 155  USD155 In stock
50mg USD 260  USD260 In stock
100mg USD 435  USD435 In stock
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Quality Control & Documentation
Biological Activity

BRL 50481 is a selective, substrate-competitive inhibitor of phosphodiesterase (PDE) 7 (Ki = 180 nM). Displays > 200-fold selectivity over PDE1B, PDE1C, PDE2, PDE3, PDE4A4 and PDE5.

Chemical Information
Molecular Weight 244.26
Formula C9H12N2O4S
CAS Number 433695-36-4
Solubility (25°C) DMSO 24.43 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Takahashi, et al. Eur J Pharmacol. Protective effects of SEA0400, a novel and selective inhibitor of the Na+/Ca2+ exchanger, on myocardial ischemia-reperfusion injuries.

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Keywords: BRL 50481 supplier, inhibitors, activators

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