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BRD7389 is a specific RSK family kinase inhibitor with IC50s of 1.5 μM, 2.4 μM, and 1.2 μM for RSK1, RSK2, and RSK3, respectively. BRD7389 is a small-molecule inducer of insulin expression in pancreatic α-cells.
| Molecular Weight | 366.41 |
| Formula | C24H18N2O2 |
| CAS Number | 376382-11-5 |
| Form | Solid |
| Solubility (25°C) | DMSO 20.83 mg/mL (ultrasonic and warming and heat to 60°C) |
| Storage | 4°C, protect from light |
[2] Huishan Zhao, et al. Anticancer Res. The Clinical Implications of RSK1-3 in Human Breast Cancer
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| Bisindolylmaleimide V
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