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BQU57

Cat. No. M20607

All AbMole products are for research use only, cannot be used for human consumption.

BQU57 Structure

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Quality Control & Documentation
Biological Activity

BQU57, a derivative of RBC8, is a selective GTPase Ral inhibitor relative to the GTPases Ras and RhoA.

Chemical Information
Molecular Weight 334.10
Formula C16H13F3N4O
CAS Number 1637739-82-2
Solubility (25°C) DMSO 66 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Katie A Thies, et al. Breast Cancer Res. The small G-protein RalA promotes progression and metastasis of triple-negative breast cancer

[2] Siddhi Inchanalkar, et al. Mol Pharm. Polymer Nanovesicle-Mediated Delivery of MLN8237 Preferentially Inhibits Aurora Kinase A To Target RalA and Anchorage-Independent Growth in Breast Cancer Cells

[3] Chao Yan, et al. Nature. Discovery and characterization of small molecules that target the GTPase Ral

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  Catalog
Abmole Inhibitor Catalog




Keywords: BQU57 supplier, ROCK, inhibitors, activators

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