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BQ-788 is a potent and selective ETB receptor antagonist with an IC50 of 1.2 nM inhibiting ET-1 binding to ETB receptor in human Girrardi heart cells. BQ-788 is an enhancer of AQP4(Aquaporin-4).
| Molecular Weight | 641.8 |
| CAS Number | 173326-37-9 |
| Solubility (25°C) | DMSO 100 mg/mL |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[2] M A A Arıcı, et al. Effects of BQ-788 on amitriptyline-induced cardiovascular toxicity
[3] Megumu Okada, et al. BQ-788, a selective endothelin ET(B) receptor antagonist
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