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BPKDi 

Cat. No. M27926

All AbMole products are for research use only, cannot be used for human consumption.

BPKDi  Structure

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Quality Control & Documentation
Biological Activity

BPKDi is a potent bipyridyl PKD inhibitor with IC50s of 1 nM, 9 nM and 1 nM for PKD1, PKD2 and PKD3, respectively. BPKDi blocks signal-dependent phosphorylation and nuclear export of class IIa HDACs in cardiomyocytes.

Chemical Information
Molecular Weight 380.49
Formula C21H28N6O
CAS Number 1201673-28-0
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] Lauren Monovich, et al. FEBS Lett. A novel kinase inhibitor establishes a predominant role for protein kinase D as a cardiac class IIa histone deacetylase kinase

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  Catalog
Abmole Inhibitor Catalog




Keywords: BPKDi  supplier, PKD, inhibitors, activators

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