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BMS-963272 

Cat. No. M28440

All AbMole products are for research use only, cannot be used for human consumption.

BMS-963272  Structure

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Quality Control & Documentation
Biological Activity

BMS-963272 is a potent, selective MGAT2 inhibitor (IC50 = 7.1 nM) for the research of metabolic disorders.

Chemical Information
Molecular Weight 525.45
Formula C24H21F6N5O2
CAS Number 1441057-15-3
Form Solid
Solubility (25°C) DMSO 250 mg/mL (ultrasonic)
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Dong Cheng, et al. Cell Metab. MGAT2 inhibitor decreases liver fibrosis and inflammation in murine NASH models and reduces body weight in human adults with obesity

[2] Huji Turdi, et al. J Med Chem. Screening Hit to Clinical Candidate: Discovery of BMS-963272, a Potent, Selective MGAT2 Inhibitor for the Treatment of Metabolic Disorders

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  Catalog
Abmole Inhibitor Catalog




Keywords: BMS-963272  supplier, Transferase, inhibitors, activators

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