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Bictegravir (GS-9883) Sodium is a novel and potent inhibitor of HIV-1 integrase, specifically targets IN strand transfer activity with an IC50 of 7.5 nM.
Molecular Weight | 473.38 |
Formula | C21H18F3N3O5.Na |
CAS Number | 1807988-02-8 |
Solubility (25°C) | DMSO 2 mg/mL |
Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[2] No authors listed. Bictegravir
[4] No authors listed. Bictegravir
[5] Vincenzo Spagnuolo, et al. Curr Opin HIV AIDS. Bictegravir
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Bictegravir
Bictegravir (GS-9883) is a novel, potent inhibitor of HIV-1 integrase with an IC50 of 7.5 nM. |
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