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BAY-390 

Cat. No. M29788

All AbMole products are for research use only, cannot be used for human consumption.

BAY-390  Structure

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Quality Control & Documentation
Biological Activity

BAY-390 is a selective, across species active and brain penetrating TRPA1 inhibitor. BAY-390 inhibits hTRPA1 FLIPR, hTRPA1 Ephys, rTRPA1 FLIPR and rDRG Ephys with IC50s of 16, 82, 63 and 35 nM, respectively. BAY-390 can be used for the research of inflammation.

Chemical Information
Molecular Weight 277.26
Formula C13H15F4NO
CAS Number 2741956-55-6
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] Stefanie Mesch, et al. J Med Chem. Discovery of BAY-390, a Selective CNS Penetrant Chemical Probe as Transient Receptor Potential Ankyrin 1 (TRPA1) Antagonist

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  Catalog
Abmole Inhibitor Catalog




Keywords: BAY-390  supplier, TRP Channel, inhibitors, activators

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