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Firmonertinib mesylate

Cat. No. M9400

All AbMole products are for research use only, cannot be used for human consumption.

Firmonertinib mesylate Structure
Synonym:

Alflutinib mesylate; AST2818 mesylate

Size Price Availability Quantity
5mg USD 215  USD215 In stock
10mg USD 320  USD320 In stock
50mg USD 900  USD900 In stock
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Quality Control & Documentation
Biological Activity

Firmonertinib (Alflutinib) mesylate is a potent, third generation EGFR inhibitor that targets both EGFR activating mutations and T790M thus leading to tumor growth inhibition. Firmonertinib (AST2818) has the potential for the research of non-small cell lung cancer (NSCLC).

Chemical Information
Molecular Weight 664.7
Formula C29H35F3N8O5S
CAS Number 2130958-55-1
Solubility (25°C) DMSO 4 mg/mL (Need ultrasonic)
Storage 4°C, dry, sealed
References

[1] Y Shi, et al. J Thorac Oncol. Third Generation EGFR Inhibitor AST2818 (Alflutinib) in NSCLC Pat-ients with EGFR T790M Mutation: A phase1/2 Multi-Center Clinical Trial.

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Keywords: Firmonertinib mesylate, Alflutinib mesylate; AST2818 mesylate supplier, EGFR/HER2, inhibitors, activators

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