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ARD-2128 is a highly potent, orally bioavailable PROTAC androgen receptor (AR) degrader. ARD-2128 effectively reduces AR protein, suppresses AR-regulated genes in tumor tissues, and inhibits growth of tumor without signs of toxicity. ARD-2128 has the potential for the research of the prostate cancer.
| Molecular Weight | 820.37 |
| Formula | C45H50ClN7O6 |
| CAS Number | 2222111-87-5 |
| Form | Solid |
| Solubility (25°C) | DMSO 100 mg/mL (ultrasonic) |
| Storage | -20°C, protect from light, dry, sealed |
| Related PROTAC Products |
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| ZXH-4-130 TFA
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| MS4322
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Products are for research use only. Not for human use. We do not sell to patients.
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