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AF-DX 116 is a selective M2 muscarinic acetylcholine receptor antagonist.
| Molecular Weight | 421.54 |
| Formula | C24H31N5O2 |
| CAS Number | 102394-31-0 |
| Form | Solid |
| Solubility (25°C) | DMSO: 5 mg/mL warmed |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[3] R Micheletti, et al. AF-DX 116, a cardioselective muscarinic antagonist
[4] H F Pitschner, et al. AF-DX 116 discriminates heart from gland M2-cholinoceptors in man
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