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Otenzepad (AF-DX 116) is a selective M2 muscarinic acetylcholine receptor antagonist.
| Molecular Weight | 421.54 |
| Formula | C24H31N5O2 |
| CAS Number | 102394-31-0 |
| Form | Solid |
| Solubility (25°C) | DMSO: 5 mg/mL warmed |
| Storage |
Powder -20°C 3 years ; 4°C 2 years In solvent -80°C 6 months ; -20°C 1 month |
[3] R Micheletti, et al. AF-DX 116, a cardioselective muscarinic antagonist
[4] H F Pitschner, et al. AF-DX 116 discriminates heart from gland M2-cholinoceptors in man
| Related AChR/AChE Products |
|---|
| Methoctramine tetrahydrochloride
Methoctramine tetrahydrochloride is a potent and cardioselectivity antagonist of M2 muscarinic receptor. |
| AT 1001
AT 1001 is a high-affinity and selective antagonist of the α3β4 nicotinic acetylcholine receptor (α3β4 nAChR) with Ki of 2.64 nM. |
| Dihydro-β-erythroidine hydrobromide
Dihydro-β-erythroidine hydrobromide is a potent, orally active, and competitive antagonist of neuronal nAChRs. Dihydro-β-erythroidine hydrobromide shows selectivity for α4β4 and α4β2 nAChRs, with IC50s of 0.19 and 0.37 μM, respectively. |
| Spinosad
Spinosad, a mixture of spinosyns A and D known as fermentation products of a soil actinomycete (Saccharopolyspora spinosa), is a biological neurotoxic insecticide with a broader action spectrum. Spinosad targets the nicotinic acetylcholine receptor (nAChRs) of the insect nervous system. |
| TAE-1
TAE-1 is a potent inhibitor of AChE and BuChE. |
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