Free shipping on all orders over $ 500

Abarelix

Cat. No. M13376

All AbMole products are for research use only, cannot be used for human consumption.

Abarelix Structure
Synonym:

R3827; PPI 149

Size Price Availability Quantity
5mg USD 74  USD74 In stock
10mg USD 115  USD115 In stock
25mg USD 240  USD240 In stock
50mg USD 380  USD380 In stock
Free Delivery on orders over USD 500 Bulk Inquiry?

Quality Control & Documentation
Biological Activity

Abarelix (R3827) is the first approved antagonist for the study of GnRH in advanced prostate cancer. Sequence:Ac-{d-2-Nal}-{d-4-Cpa}-{d-3-Pal}-S-{NMyr}-{d-Asp}-L-K(ipr)-P-{d-Ala}-NH2

Chemical Information
Molecular Weight 1416.06
Formula C72H95ClN14O14
CAS Number 183552-38-7
Form Solid
Solubility (25°C) DMSO : ≥ 14.2 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] Roger S Kirby, et al. BJU Int. Abarelix and other gonadotrophin-releasing hormone antagonists in prostate cancer

[2] Frans Debruyne, et al. Future Oncol. Abarelix for injectable suspension: first-in-class gonadotropin-releasing hormone antagonist for prostate cancer

[3] William P Hogle. Clin J Oncol Nurs. Abarelix (plenaxis)

[4] Pierre Mongiat-Artus, et al. Expert Opin Pharmacother. Abarelix: the first gonadotrophin-releasing hormone antagonist for the treatment of prostate cancer

[5] No authors listed. Drugs R D. Abarelix: abarelix-depot-F, abarelix-depot-M, abarelix-L, PPI 149, R 3827

Related LHRH/GnRH Products
GnRH antagonist 2 

GnRH antagonist 2 (formula I) is a GnRH receptor antagonist that can be used for endometriosis research.

Kisspeptin-54(human)

Kisspeptin-54(human) (Metastin(human)) is an endogenous ligand for kisspeptin receptor (KISS1, GPR54).

Luteinizing Hormone Releasing Hormone (LH-RH), salmon

Luteinizing Hormone Releasing Hormone (LH-RH), salmon (Salmon GnRH) is the hypophysiotropic decapeptide synthesized in the hypothalamus that plays a crucial role in the control of reproductive functions.

Phoenixin-14

Phoenixin-14 (PNX-14) is one of the endogenous active isoform, and generates anxiolytic effect via the activation of the AHA GnRH system in mice.

LGnRH-III, lamprey

LGnRH-III, lamprey, an isoform of GnRH isolated from the sea lamprey, is a weak GnRH agonist with antitumor activities.

  Catalog
Abmole Inhibitor Catalog




Keywords: Abarelix, R3827; PPI 149 supplier, LHRH/GnRH, inhibitors, activators

All AbMole products are for research use only, cannot be used for human consumption or veterinary use. We do not provide products or services to individuals. Please comply with the intended use and do not use AbMole products for any other purpose.



Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2024 AbMole BioScience. All Rights Reserved.