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2-Methoxyestrone

Cat. No. M14345

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2-Methoxyestrone Structure
Size Price Availability Quantity
1mg USD 60  USD60 In stock
5mg USD 150  USD150 In stock
10mg USD 240  USD240 In stock
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Quality Control & Documentation
Biological Activity

2-Methoxyestrone is a methoxylated catechol estrogen and metabolite of estrone, with a pKa of 10.81.

Chemical Information
Molecular Weight 300.39
CAS Number 362-08-3
Solubility (25°C) DMSO 50 mg/mL
Storage Powder          -20°C   3 years ;  4°C   2 years
In solvent       -80°C   6 months ;  -20°C   1 month
References

[1] R HOBKIRK, et al. 2-methoxyestrone as an estrogen metabolite in the human subject

[2] A Singh, et al. Inhibition of deoxyglucose uptake in MCF-7 breast cancer cells by 2-methoxyestrone and 2-methoxyestrone-3-O-sulfamate

[3] C Longcope, et al. Metabolism of 2-methoxyestrone in normal men

[4] C P Martucci. The role of 2-methoxyestrone in estrogen action

[5] P Ball, et al. Radioimmunoassay of 2-hydroxyesterone and 2-methoxyestrone in human urine

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Keywords: 2-Methoxyestrone supplier, Metabolite/Endogenous Metabolite, inhibitors, activators

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