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ST4206 

Cat. No. M28033

All AbMole products are for research use only, cannot be used for human consumption.

ST4206  Structure

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Quality Control & Documentation
Biological Activity

ST4206 is a potent and orally active adenosine A2A receptor antagonist, with Kis of 12 nM and 197 nM for adenosine A2A receptor and adenosine A1 receptor, respectively. ST4206 has the potential for Parkinson׳s disease research.

Chemical Information
Molecular Weight 286.29
Formula C12H14N8O
CAS Number 1246018-36-9
Storage Please store the product under the recommended conditions in the Certificate of Analysis.
References

[1] Maria Antonietta Stasi, et al. Eur J Pharmacol. Animal models of Parkinson׳s disease: Effects of two adenosine A2A receptor antagonists ST4206 and ST3932, metabolites of 2-n-Butyl-9-methyl-8-[1,2,3]triazol-2-yl-9H-purin-6-ylamine (ST1535)

[2] Annalisa Pinna. CNS Drugs. Adenosine A2A receptor antagonists in Parkinson's disease: progress in clinical trials from the newly approved istradefylline to drugs in early development and those already discontinued

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Abmole Inhibitor Catalog




Keywords: ST4206  supplier, Adenosine Receptor, inhibitors, activators

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