Glutaminase Glutaminase

Inhibitor

Cat.No.	Name	Information
M10745	6-Diazo-5-oxo-L-norleucine	6-Diazo-5-oxo-L-norleucine (Diazooxonorleucine, L-6-Diazo-5-oxonorleucine, DON) is an antibiotic isolated from Streptomyces, an antagonist of glutaminase with an IC50 value of about 1 mM for cKGA (renal glutamine). 6-Diazo-5-oxo-L-norleucine has analgesic, antibacterial, antiviral and anti-cancer properties.
M9215	GK921	GK921 is a transglutaminase 2 (TGase 2) inhibitor.
M6285	Glutaminase C-IN-1	Glutaminase C-IN-1 (Compound 968) is an allosteric inhibitor of Glutaminase C that inhibits cancer cell growth without affecting their normal cellular counterparts.
M5015	BPTES	BPTES is a potent and selective Glutaminase GLS1 (KGA) inhibitor with IC50 of 0.16 μM.
M52577	2-Amino-2-(p-tolyl)acetic acid	2-Amino-2-(p-tolyl)acetic acid is used for optimizing azide skeleton, and is the intermediate in the synthesis of 1,3, 4-thiadiazole compounds.
M42427	BJJF078	BJJF078 is an aminopiperidine derivative.
M42426	TG53	TG53 is a potent inhibitor of tissue transglutaminase (TG2) and fibronectin (FN) protein-protein interaction.
M42425	GLS1 Inhibitor-7	GLS1 Inhibitor-7 is a GLS1 inhibitor (IC50=46.7 μM), with potential anti-cancer, anti-aging and anti-obesity properties.
M28224	NC9	NC9 (Cbz-Lys(Acr)-PEG2-dansyl) is an irreversible transglutaminase (TG) inhibitor. NC9 inhibits osteoblast differentiation and mineralization. NC9 destabilizes microtubules. NC9 can be used for the research of osteoblast differentiation.