Inhibitor
| Cat.No. | Name | Information |
|---|---|---|
| M20875 | L-Albizziin | L-albizziin (L-alpha-amino-beta-ureidopropionic acid) is a potent inhibitor of glutamase. L-albizziin interferes with the utilisation of L-glutamine by the Debaryomyces spp. enzyme probably in a competitive and reversible manner since L-albizziin is also a substrate of the enzyme. |
| M10745 | 6-Diazo-5-oxo-L-norleucine | 6-Diazo-5-oxo-L-norleucine (Diazooxonorleucine, L-6-Diazo-5-oxonorleucine, DON) is an antibiotic isolated from Streptomyces, an antagonist of glutaminase with an IC50 value of about 1 mM for cKGA (renal glutamine). 6-Diazo-5-oxo-L-norleucine has analgesic, antibacterial, antiviral and anti-cancer properties. |
| M9215 | GK921 | GK921 is a transglutaminase 2 (TGase 2) inhibitor. |
| M6285 | Glutaminase C-IN-1 | Glutaminase C-IN-1 (Compound 968) is an allosteric inhibitor of Glutaminase C that inhibits cancer cell growth without affecting their normal cellular counterparts. |
| M5015 | BPTES | BPTES is a potent and selective Glutaminase GLS1 (KGA) inhibitor with IC50 of 0.16 μM. |
| M56697 | ZED-1227 | ZED-1227 is a specific and orally active transglutaminase 2 (TG2) inhibitor, with an IC50 of 45 nM. |
| M56696 | TG-2-IN-1 | TG-2-IN-1 is a transglutaminase-2 (TGM-2) inhibitor. |
| M52577 | 2-Amino-2-(p-tolyl)acetic acid | 2-Amino-2-(p-tolyl)acetic acid is used for optimizing azide skeleton, and is the intermediate in the synthesis of 1,3, 4-thiadiazole compounds. |
| M42427 | BJJF078 | BJJF078 is an aminopiperidine derivative. |
| M42426 | TG53 | TG53 is a potent inhibitor of tissue transglutaminase (TG2) and fibronectin (FN) protein-protein interaction. |
| M42425 | GLS1 Inhibitor-7 | GLS1 Inhibitor-7 is a GLS1 inhibitor (IC50=46.7 μM), with potential anti-cancer, anti-aging and anti-obesity properties. |
| M28224 | NC9 | NC9 (Cbz-Lys(Acr)-PEG2-dansyl) is an irreversible transglutaminase (TG) inhibitor. NC9 inhibits osteoblast differentiation and mineralization. NC9 destabilizes microtubules. NC9 can be used for the research of osteoblast differentiation. |
| M10836 | IPN60090 | IPN-60090 (IACS-6274) is an inhibitor of orally active and highly selective glutaminease 1 GLS1 (IC50=31 nM), inactive against GLS-2. IPN-60090 (IACS-6274) exhibits excellent physicochemical and pharmacokinetic properties in vivo. IPN-60090 can be used in the study of solid tumors such as lung and ovarian cancers. |
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