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Ephrin Receptor Eph receptor tyrosine kinase (RTK)

Inhibitor

Cat.No.  Name Information
M8974 ALW-II-41-27 ALW-II-41-27 is a Eph receptor tyrosine kinase inhibitor with an IC50 of 11 nM for EPHA2.
M49948 KYL peptide KYL peptide is an antagonistic peptide that selectively targets EphA4, and its binding to the ligand-binding domain of EphA4 effectively alleviates Aβ-induced synaptic dysfunction and synaptic plasticity defects in AD mice. In addition, KYL peptide can promote nerve regeneration after injury and modulate immune response.
M43494 Eph inhibitor 1 Eph inhibitor 1 is a potent Eph inhibitor.
M43493 Urolithin D Urolithin D is competitive and reversible antagonist of EphA receptors.
M29119 123C4  123C4 is a potent, selective and competitive agonist of the receptor tyrosine kinase EPHA4, with a Ki value of 0.65 μM.
M27828 ALW-II-49-7  ALW-II-49-7 is a selective EphB2 kinase inhibitor with an EC50 value of 40 nM in cell.
M14892 NVP-BHG712 isomer NVP-BHG712 isomer, a regioisomer of NVP-BHG712, shows conserved non-bonded binding to EPHA2 and EPHB4.
M49950 EphA2 agonist 1 EphA2 agonist 1 is a potent EphA2 receptor agonist.EphA2 agonist 1 is highly active and selective for EphA2 overexpressing glioma cells and stimulates EphA2 phosphorylation.
M49949 LDN-211904 oxalate LDN-211904 oxalate is a potent and selective EphB3 inhibitor with an IC50 of 0.079 µM.LDN-211904 oxalate showed good metabolic stability in mouse liver microsomes.LDN-211904 oxalate was shown to be effective in inhibiting STAT3-activated CSC stemness in combination with cetuximab.
M49947 Ifabotuzumab Ifabotuzumab is an IgG1κ antibody (KD=610 pM) targeting EphA3. Ifabotuzumab is able to cause apoptosis of tumor cells and activate antibody-dependent cell-mediated cytotoxicity (ADCC), which disrupts the tumor vascular system. In addition, Ifabotuzumab reduces idiopathic pulmonary fibrosis (IPF) CCR10+ cells and ameliorates pulmonary fibrosis.
M28752 UniPR129  UniPR129 is a potent Eph/ephrin antagonist. UniPR129 has the potential for the research of cancer disease.
M20738 Eph-inhibitor-1 Eph-inhibitor-1 (Eph inhibitor 2) is an Eph family tyrosine kinase inhibitor that targets Eph receptors.




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