Catalog

CGRP Receptor Calcitonin gene-related peptide Receptor

Inhibitors

Cat.No.	Name	Information
M10372	Vazegepant hydrochloride	Vazegepant (BHV-3500) hydrochloride is a highly affinity CGRP receptor antagonist (hCGRP Ki= 0.023 nM).
M9165	Rimegepant	Rimegepant, also known as BMS-927711, is a potent, selective, competitive, and orally active calcitonin gene-related peptide (CGRP) antagonist with a Ki value of 0.027 nM.
M5223	BAR501	BAR501 is a potent and selective agonist of GPBAR1 with an EC50 of 1 μM.
M3618	MK-0974	MK-0974 (Telcagepant) is a highly potent, selective and orally bioavailable CGRP receptor antagonist with Ki values of 0.77 nM and 1.2 nM for human and rhesus CGRP receptors respectively.
M2133	MK-3207 hydrochloride	MK-3207 hydrochloride is a potent CGRP receptor antagonist with IC50 of 0.12 nM.