Inhibitors
Cat.No. | Name | Information |
---|---|---|
M10894 | Ubrogepant | Ubrogepant (MK-1602) is a novel oral calcitonin gene-associated peptide receptor (CGRP) antagonist with the potential to be used in acute migraine studies. |
M10801 | Calcitonin (salmon) | Calcitonin salmon is a calcium-regulating hormone that is a dual agonist of amylin and calcitonin receptors that stimulate bone production and inhibit bone resorption. |
M10372 | Vazegepant hydrochloride | Vazegepant (BHV-3500) hydrochloride is a highly affinity CGRP receptor antagonist (hCGRP Ki= 0.023 nM). |
M9165 | Rimegepant | Rimegepant, also known as BMS-927711, is a potent, selective, competitive, and orally active calcitonin gene-related peptide (CGRP) antagonist with a Ki value of 0.027 nM. |
M6504 | Olcegepant (BIBN-4096) | Olcegepant (BIBN-4096) is a potent and selective non-peptide antagonist of the calcitonin gene-related peptide (CGRP) receptor with IC50 of 0.03 nM and Ki of 14.4 pM for human CGRP. |
M5223 | BAR501 | BAR501 is a potent and selective agonist of GPBAR1 with an EC50 of 1 μM. |
M3618 | MK-0974 | MK-0974 (Telcagepant) is a highly potent, selective and orally bioavailable CGRP receptor antagonist with Ki values of 0.77 nM and 1.2 nM for human and rhesus CGRP receptors respectively. |
M2133 | MK-3207 hydrochloride | MK-3207 hydrochloride is a potent CGRP receptor antagonist with IC50 of 0.12 nM. |
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