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CGRP Receptor Calcitonin gene-related peptide Receptor

Inhibitors

Cat.No.  Name Information
M10894 Ubrogepant Ubrogepant (MK-1602) is a novel oral calcitonin gene-associated peptide receptor (CGRP) antagonist with the potential to be used in acute migraine studies.
M10801 Calcitonin (salmon) Calcitonin salmon is a calcium-regulating hormone that is a dual agonist of amylin and calcitonin receptors that stimulate bone production and inhibit bone resorption.
M10372 Vazegepant hydrochloride Vazegepant (BHV-3500) hydrochloride is a highly affinity CGRP receptor antagonist (hCGRP Ki= 0.023 nM).
M9165 Rimegepant Rimegepant, also known as BMS-927711, is a potent, selective, competitive, and orally active calcitonin gene-related peptide (CGRP) antagonist with a Ki value of 0.027 nM.
M6504 Olcegepant (BIBN-4096) Olcegepant (BIBN-4096) is a potent and selective non-peptide antagonist of the calcitonin gene-related peptide (CGRP) receptor with IC50 of 0.03 nM and Ki of 14.4 pM for human CGRP.
M5223 BAR501 BAR501 is a potent and selective agonist of GPBAR1 with an EC50 of 1 μM.
M3618 MK-0974 MK-0974 (Telcagepant) is a highly potent, selective and orally bioavailable CGRP receptor antagonist with Ki values of 0.77 nM and 1.2 nM for human and rhesus CGRP receptors respectively.
M2133 MK-3207 hydrochloride MK-3207 hydrochloride is a potent CGRP receptor antagonist with IC50 of 0.12 nM.



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