|M10894||Ubrogepant||Ubrogepant (MK-1602) is a novel oral calcitonin gene-associated peptide receptor (CGRP) antagonist with the potential to be used in acute migraine studies.|
|M10801||Calcitonin (salmon)||Calcitonin salmon is a calcium-regulating hormone that is a dual agonist of amylin and calcitonin receptors that stimulate bone production and inhibit bone resorption.|
|M10372||Vazegepant hydrochloride||Vazegepant (BHV-3500) hydrochloride is a highly affinity CGRP receptor antagonist (hCGRP Ki= 0.023 nM).|
|M9165||Rimegepant||Rimegepant, also known as BMS-927711, is a potent, selective, competitive, and orally active calcitonin gene-related peptide (CGRP) antagonist with a Ki value of 0.027 nM.|
|M6504||Olcegepant (BIBN-4096)||Olcegepant (BIBN-4096) is a potent and selective non-peptide antagonist of the calcitonin gene-related peptide (CGRP) receptor with IC50 of 0.03 nM and Ki of 14.4 pM for human CGRP.|
|M5223||BAR501||BAR501 is a potent and selective agonist of GPBAR1 with an EC50 of 1 μM.|
|M3618||MK-0974||MK-0974 (Telcagepant) is a highly potent, selective and orally bioavailable CGRP receptor antagonist with Ki values of 0.77 nM and 1.2 nM for human and rhesus CGRP receptors respectively.|
|M2133||MK-3207 hydrochloride||MK-3207 hydrochloride is a potent CGRP receptor antagonist with IC50 of 0.12 nM.|
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