About 1 result found for searched term "Vicriviroc maleate" (0.714 seconds)
Cat.No. | Name | Target |
---|---|---|
M30343 | Vicriviroc maleate | CCR |
SCH-417690 maleate; SCH-D maleate | ||
Vicriviroc maleate (SCH-417690 maleate; SCH-D maleate) is a potent, selective, oral bioavailable and CNS penetrated antagonist of CCR5, with a Ki of 2.5 nM, and also inhibits HIV-1 in PBMC cells, with IC90s of 3.3 nM (JrFL), 2.8 nM (ADA-M), 1.8 nM (301657), 4.9 nM (JV1083) and 10 nM (RU 570). |
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