About 4 results found for searched term "Varenicline" (0.077 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M6268 | Varenicline | AChR/AChE |
| CP 526555 | ||
| Varenicline (CP 526555) is a selective α4β2 nicotinic receptor partial agonist, it stimulates nicotine receptors more weakly than nicotine itself does. | ||
| M6273 | Varenicline tartrate | AChR/AChE |
| CP 526555-18 | ||
| Varenicline Tartrate is a nicotinic AChR partial agonist, used to treat nicotine addiction. | ||
| M9058 | Varenicline hydrochloride | AChR/AChE |
| CP 526555 hcl; Chantix; Champix | ||
| Varenicline hydrochloride is a potent partial agonist of α4β2 nicotinic acetylcholine receptor (nAChR) and α3β4 nAChR, with EC50s of 2.3 μM and 55 μM, respectively. In addition, Varenicline hydrochloride is also a potent full agonist of α7 nAChRs. In addition, Varenicline hydrochloride is a potent full α7 nAChRs agonist with an EC50 of 18 μM. | ||
| M20984 | Varenicline dihydrochloride | AChR/AChE |
| Chantix, Champix | ||
| Varenicline (CP 526555, Chantix, Champix) dihydrochloride is a potent, partial agonist of α4β2 nicotinic acetylcholine receptor (nAChR) and α3β4 nAChR with EC50 of 2.3 μM and 55 μM, respectively. Varenicline dihydrochloride is a potent, full agonist of α7 nAChRs with EC50 of 18 μM. Varenicline is a prescription medication used for smoking cessation. | ||
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