TRAP-7 - Search Results | AbMole BioScience

About 7 results found for searched term "TRAP-7" (0.131 seconds)

Cat.No.	Name	Target
M52912	TRAP-7	PAR
	TRAP-7 is a thrombin receptor (PAR) activating peptide.
M2142	Anacetrapib	CETP
	MK-0859
	Anacetrapib is an orally active and potent inhibitor of CETP with IC50 of 7.9 nM and 11.8 nM for rhCETP and mutant CETP(C13S) respectively.
M3438	Dalcetrapib	CETP
	JTT-705, RO4607381
	Dalcetrapib (JTT-705) is a rhCETP inhibitor with IC50 of 0.2 μM that increases the plasma HDL cholesterol.
M9771	TRAP-6	Peptides
	Thrombin Receptor Activator Peptide 6; PAR-1 agonist peptide
	TRAP-6 (Thrombin Receptor Activator Peptide 6) is a peptide fragment (residues 42-47) of protease-activated receptor 1 (PAR1) that acts as a PAR1 agonist.
M20676	Pimitespib	HSP
	TAS-116
	TAS-116 is a novel, small-molecule HSP90 inhibitor which inhibits geldanamycin-FITC binding to HSP90 proteins with Ki values of 34.7 nmol/L, 21.3 nmol/L, >50,000 nmol/L, and >50,000 nmol/L for HSP90α, HSP90β, GRP94, and TRAP1, respectively. Furthermore, TAS-116 does not inhibit other ATPases such as HSP70 (IC50 >200 μmol/L).
M31376	DN401	HSP
	DN401 is a potent TRAP1 and Hsp90 inhibitor with anticancer activity with IC50 values of 79 nM and 698 nM, respectively.
M53841	Ac-YVAD-CHO	IL Receptor/Related
	Ac-YVAD-CHO (L-709049) is a potent, reversible, specific tetrapeptide interleukin-lβ converting enzyme (ICE) inhibitor with mouse and human Ki values of 3.0 and 0.76 nM.