About 3 results found for searched term "SIK2-IN-1" (0.132 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M42053 | SIK2-IN-1 | Salt-inducible Kinase |
| SIK2-IN-1 is a potent SIK2 inhibitor over other AMPK kinases. | ||
| M11237 | ARN-3236 | Salt-inducible Kinase |
| Arn-3236 is a selective inhibitor of salt-induced kinase 2 (SIK2) with an IC50 value of <1 nM, 21.63 nM and 6.63 nM against SIK2, SIK1 and SIK3, respectively. It has antitumor activity. | ||
| M28491 | MRT199665 | Salt-inducible Kinase |
| MRT199665 is a potent and ATP-competitive, selective MARK/SIK/AMPK inhibitor with IC50s of 2/2/3/2 nM, 10/10 nM, and 110/12/43 nM for MARK1/MARK2/MARK3/MARK14, AMPKα1/AMPKα2, and SIK1/SIK2/SIK3, respectively. MRT199665 causes apoptosis in MEF2C-activated human acute myeloid leukemias (AML) cells. MRT199665 inhibits the phosphorylation of SIK substrate CRTC3 at S370. | ||
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