HIV-1 protease-IN-3 - Search Results

About 6 results found for searched term "HIV-1 protease-IN-3" (0.14 seconds)

Cat.No.	Name	Target
M41183	HIV-1 protease-IN-3	Anti-infection
	HIV-1 protease-IN-3 is a potent inhibitor of HIV-1 protease (IC50=71 nM; EC50=0.86 μM).
M1657	Atazanavir Sulfate	HIV Protease
	BMS-232632, Reyataz, CGP-73547
	Atazanavir sulfate (BMS-232632, Reyataz) is an azapeptide inhibitor of HIV-1 protease. Atazanavir sulfate is a substrate and inhibitor of CYP3A4, and an inhibitor and inducer of P-glycoprotein (P-gp). Atazanavir sulfate is also a SARS-CoV 3CLpro inhibitor with an IC50 of 3.49 μM.
M27589	TMC310911	HIV Protease
	ASC-09
	TMC310911 is a potent and orally active HIV type-1 (HIV-1) protease inhibitor with EC50 values ranged from 2.2 nM to 14.2 nM for wild-type HIV-1. TMC310911 has potent activity against a wide spectrum of recombinant HIV-1 isolates. TMC310911 has strong antiviral activity.
M38764	Indinavir	Anti-infection
	Indinavir (MK-639 free base) is an orally active and selective HIV-1 protease inhibitor with a Ki of 0.54 nM for PR. Indinavir exhibits anticancer activity by inhibiting the activation of MMPs-2 hydrolysis, anti-angiogenesis and inducing apoptosis. Indinavir is also a SARS-CoV 3CLpro inhibitor.
M41192	HIV-1 protease-IN-8	HIV Protease
	HIV-1 protease-IN-8 is a potent HIV-1 protease inhibitor with an IC50 value of 0.32 nM.
M53461	HIV-1 protease-IN-7	HIV Protease
	HIV-1 protease-IN-7 is an orally active HIV-1 protease inhibitor (IC50=3.52 nM, EC50=37 nM).