About 5 results found for searched term "EZH2-IN-15" (0.129 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M41699 | EZH2-IN-15 | Histone Methyltransferase |
| EZH2-IN-15 (SHR2554) is a EZH2 inhibitor. | ||
| M2676 | EPZ005687 | EZH2 |
| EPZ005687 is a potent, selective EZH2 inhibitor,Ki The value is 24 nM, which is 50 times more selective than EZH1 and 500 times more selective than 15 other methyltransferases. | ||
| M11242 | EI1 | Histone Methyltransferase |
| KB-145943 | ||
| EI1 (KB-145943) is a novel and effective EZH2 inhibitor, capable of acting on EZH2 (WT) and EZH2 (Y641F) with IC50 values of 15 nM and 13 nM, respectively. | ||
| M13846 | EPZ011989 trifluoroacetate | Histone Methyltransferase |
| EPZ-011989 trifluoroacetate | ||
| EPZ011989 trifluoroacetate is a potent, selective orally bioavailable EZH2 inhibitor with Ki < 3 nM for EZH2 wt and EZH2 Y646; 15-fold selectivity over EZH1 and >3000-fold selectivity over other HMTase. | ||
| M28933 | ZLD1039 | Histone Methyltransferase |
| ZLD1039 is a potent, highly selective, and orally bioavailable EZH2 inhibitor. ZLD1039 shows potent and concentration-dependent inhibition of PRC2 enzymatic activity against EZH2 wild-type as well as Y641F, and A677G mutant enzymes with IC50 values of 5.6, 15, and 4.0 nM, respectively. ZLD1039 inhibits breast tumor growth and metastasis. | ||
Products are for research use only. Not for human use. We do not sell to patients.
© Copyright 2010-2023 AbMole BioScience. All Rights Reserved.
