About 9 results found for searched term "58-49-1" (0.131 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M29719 | Anrikefon acetate | Opioid Receptor |
| HSK21542 acetate | ||
| Anrikefon (HSK21542) acetate is a kappa opioid receptor agonist with analgesic effect. | ||
| M30325 | Angiotensin II 5-valine | Angiotensin Receptor |
| Valine angiotensin II; 5-L-Valine angiotensin II | ||
| Angiotensin II 5-valine is an agonist of angiotensin receptor. | ||
| M42276 | MK 386 | Others |
| MK 386 (L-733692) is a selective 5-α-reductase I inhibitor, used for prostate cancer inhibition. | ||
| M44639 | N-trans-p-Coumaroyl-N'-trans-feruloyl-3-hydroxy-cadaverine | Others |
| N-trans-p-Coumaroyl-N'-trans-feruloyl-3-hydroxy-cadaverine | ||
| M9160 | BMS-582949 | p38 MAPK |
| PS540446; BMS582949 free base | ||
| BMS-582949 is a potent and selective P38 mitogen-activated protein kinase (P38 MAPK) inhibitor with IC50 of 13nM. | ||
| M25541 | SKF-82958 hydrobromide | Dopamine Receptor |
| (±)-SKF-82958 hydrobromide; Chloro-APB hydrobromide | ||
| SKF-82958 ((±)-SKF 82958) hydrobromide is a dopamine D1 receptor full agonist (K0.5=4 nM), displays selective for D1 over D2 receptors (K0.5=73 nM). SKF-82958 hydrobromide induces dopamine D1 receptor-dependent adenylate cyclase activity in rat striatal membranes (EC50=491 nM). | ||
| M14174 | BMS-582949 hydrochloride | p38 MAPK |
| BMS-582949 hydrochloride is an orally active and highly selective p38α MAPK inhibitor, with an IC50 of 13 nM. BMS-582949 hydrochloride displays a significantly improved pharmacokinetic profile and is effective in inflammatory disease. | ||
| M28632 | CMF019 | Others |
| CMF019 is a potent and small molecule agonist at Apelin receptor (APJ) with G protein bias. CMF019 binds to APJ with pKi values of 8.58, 8.49 and 8.71 for human, rat, and mouse, respectively. CMF019 mimics the beneficial cardiovascular actions of apelin in rodents. Apelin receptor (APJ) is a G protein-coupled receptor (GPCR) activated by the endogenous peptide apelin. | ||
| M30865 | NSC-658497 | Ras |
| NSC-658497 is an effective inhibitor of Ras-GEF, SOS1. NSC-658497 binds to SOS1, competitively suppresses SOS1-Ras interaction, and dose-dependently inhibits SOS1 GEF activity. NSC-658497 showed dose-dependent efficacy in inhibiting Ras, downstream signaling activities, and associated cell proliferation. | ||
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