About 2 results found for searched term "566-65-4" (0.209 seconds)
Cat.No. | Name | Target |
---|---|---|
M59095 | 5α-Dihydroprogesterone | Metabolite/Endogenous Metabolite |
5α-Pregnane-3,20-dione; 5-alpha-Dihydroprogesterone | ||
5α-Dihydroprogesterone (5a-Pregnane-3,20-dione) is the endogenous progesterone metabolite. 5α-Dihydroprogesterone (5a-Pregnane-3,20-dione) decreases cell-substrate attachment, adhesion plaques, vinculin expression, and polymerizes F-actin in MCF-7 breast cancer cells. | ||
M30801 | KPT-6566 | Others |
KPT-6566 is a selective and covalent prolyl isomerase PIN1 inhibitor, covalently binds to the catalytic site of PIN1, selectively inhibits and degrades PIN1. KPT-6566 shows an IC50 value of 640 nM and a Ki value of 625.2 nM for PIN1 PPIase domain. KPT-6566 can be used for the research of cancer. |
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