About 11 results found for searched term "52-49-3" (0.055 seconds)
| Cat.No. | Name | Target |
|---|---|---|
| M6032 | Trihexyphenidyl hydrochloride | AChR/AChE |
| Benzhexol hydrochloride, Artane hydrochloride | ||
| Trihexyphenidyl hydrochloride is a potent and selective M1 muscarinic receptor antagonist. Trihexyphenidyl hydrochloride shows anticholinergic activity. | ||
| M7744 | Dihydrokainic acid | GLUT |
| Dihydrokainic acid is a selective inhibitor of the GLT-1 glutamate transporter. | ||
| M10515 | JNJ-10229570 | Melanocortin Receptor |
| UNII-N9IX402L35; JNJ10229570 | ||
| JNJ-10229570 (UNII-N9IX402L35) is is a novel MC1R and MC5R antagonist, which inhibits the binding of 125I-NDP-α-MSH to cells expressing human MC1R and MC5R with IC50 values of 270 nM and 200 nM, respectively. | ||
| M11206 | A-317491 | P2 Receptor |
| A-317491 is a potent, selective and non-nucleotide antagonist of P2X3 and P2X2/3 receptors, with Kis of 22, 22, 9, and 92 nM for hP2X3, rP2X3, hP2X2/3, and rP2X2/3, respectively. A-317491 is highly selective for other P2 receptors and neurotransmitter receptors, ion channels, and enzymes (IC50>10 μM). | ||
| M14245 | A-317491 sodium salt hydrate | P2 Receptor |
| A-317491 sodium salt hydrate is a potent, selective and non-nucleotide antagonist of P2X3 and P2X2/3 receptors, with Kis of 22, 22, 9, and 92 nM for hP2X3, rP2X3, hP2X2/3, and rP2X2/3, respectively. | ||
| M19448 | Ajugol | Parasite |
| Ajugol is an iridoid glycoside that can be isolated from Leonurus artemisia. Ajugol has anti-protozoal activity againt Trypanosoma b. rhodesiense with an IC50 of 31.8 μg/mL. | ||
| M28949 | (Rac)-MGV354 | Guanylate Cyclase |
| (Rac)-MGV354 is the racemate of MGV354. MGV354 is a soluble guanylate cyclase (sGC) activator with EC50s of <0.5 nM, and 5 nM in CHO and GTM-3 E cells, respectively. | ||
| M30242 | Methoxy-PEPy | GluR |
| Methoxy-PEPy is a potent and highly selective mGlu5 receptor antagonist with IC50 of 1 nM. IC50 value: 1 nM [1] Target: mGlu5R inhibitor Administration of [3H]methoxy-PEPy (50 microCi/kg i.v.) to mGlu5 receptor-deficient mice revealed binding at background levels in forebrain, whereas wild-type mice exhibited 14-fold higher binding in forebrain relative to cerebellum . The calcium transients stimulated by these agonists were potently inhibited by reference allosteric mGlu5 antagonists - 2-methyl-6-(phenylethynyl)pyridine (MPEP), 3-[(2-methyl-1,3-thiazol-4-yl)ethynyl]pyridine (MTEP) and 3-methoxy-5-(pyridine-2-ylethynyl)pyridine (methoxy-PEPy) (IC(50) ranges: 0.8-66 nM) . | ||
| M39351 | Boc-N-methyl-L-isoleucine | Amino Acid Derivatives |
| Boc-N-methyl-L-isoleucine (Boc-N-Me-Ile-OH) is a peptide products and can be used as a precursor in organic synthesis and pharmaceuticals. | ||
| M44069 | Peonidin-3-O-arabinoside chloride | Others |
| Peonidin-3-O-arabinoside chloride | ||
| M54585 | VK-0214 | Thyroid Hormone Receptor |
| VK-0214 is an orally active, selective small molecule agonist of the thyroid receptor (THR-β) for studies related to X-linked adrenoleukodystrophy (X-ALD) and hyperlipidemia. | ||
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